Glibenclamide

• Supplier: Tocris Bioscience
• Catalog: 5133
• Prices: $65.00
• Sizes: 100 mg
• Function Type: Blocker
• Cas Number: 10238-21-8
• Chemical Name: 5-Chloro-N-[2-[4-[[[(Cylcohexylamino)carbonyl]amino]sulphonyl]phenyl]ethyl]-2-methoxybenzamide
• Formula: C23H28ClN3O5S
• Molecular Weight: 494
• Purity: >99 %
• Description: ATP-dependent K + channel (K ir 6, K ATP ) and CFTR Cl - channel blocker. Inhibits K ir 6 currents in the pancreas, causing an increase in intracellular Ca 2+ and insulin secretion. Inhibits recombinant CFTR Cl- channels with an IC 50 of 20 μ M.

Product References

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