GR 94800

Name GR 94800
Supplier Tocris Bioscience
Catalog 1483
Prices $405.00
Sizes 1 mg
Function Type Antagonist
Cas Number 141636-65-9
Formula C49H61N9O8
Molecular Weight 904.08
Description Potent and selective tachykinin NK 2 receptor antagonist (pK B values are 9.6, 6.4 and 6.0 for NK 2 , NK 1 and NK 3 receptors respectively). Active in vivo .
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Product References

Highly potent and selective heptapeptide antagonists of the neurokinin NK-2 - Highly potent and selective heptapeptide antagonists of the neurokinin NK-2

McElroy AB, Clegg SP, Deal MJ, Ewan GB, Hagan RM, Ireland SJ, Jordan CC, Porter B, Ross BC, Ward P, et al.. J Med Chem. 1992 Jul 10;35(14):2582-91.

Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic - Evidence that tachykinin NK1 and NK2 receptors mediate non-adrenergic

Zagorodnyuk V, Santicioli P, Maggi CA, Giachetti A. Br J Pharmacol. 1995 May;115(2):237-46.

An investigation of tachykinin NK2 receptor subtypes in the rat. - An investigation of tachykinin NK2 receptor subtypes in the rat.

Matuszek MA, Zeng XP, Strigas J, Burcher E. Eur J Pharmacol. 1998 Jul 3;352(1):103-9.