| Name | GSK 0660 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4918 |
| Prices | $189.00, $765.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 1014691-61-2 |
| Chemical Name | 3-[[[2-Methoxy-4-(phenylamino)phenyl]amino]sulfonyl]-2-thiophenecarboxylicacidmethylester |
| Formula | C19H18N2O5S2 |
| Molecular Weight | 418.49 |
| Purity | >99 % |
| Description | Selective PPAR δ antagonist (IC 50 values are 0.155, > 10 and ≥ 10 μ M at PPAR δ , PPAR α and PPAR γ respectively). Exhibits inverse agonist effects when administered by itself. |
| Supplier Page | Shop |
Shearer BG, Steger DJ, Way JM, Stanley TB, Lobe DC, Grillot DA, Iannone MA, Lazar MA, Willson TM, Billin AN. Mol Endocrinol. 2008 Feb;22(2):523-9. Epub 2007 Nov 1.
Wang N. PPAR Res. 2008;2008:164163.