Name | GSK 2194069 |
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Supplier | Tocris Bioscience |
Catalog | 5106 |
Prices | $235.00, $965.00 |
Sizes | 10 mg, 50 mg |
Function Type | Inhibitor |
Cas Number | 1332331-08-4 |
Chemical Name | 4-[4-(5-Benzofuranyl)phenyl]-5-[[(3S)-1-(cyclopropylcarbonyl)-3-pyrrolidinyl]methyl]-2,4-dihydro-3H-1,2,4-triazol-3-one |
Formula | C25H24N4O3 |
Molecular Weight | 428.48 |
Purity | >99 % |
Description | Potent human fatty acid synthase (hFASN) inhibitor (IC 50 = 7.7 nM); inhibits hFAS β -ketoacyl reductase activity. Inhibits lipid synthesis and attenuates proliferation of A549 non-small-cell lung cancer cells (EC 50 = 15 nM) in vitro . |
Supplier Page | Shop |