| Name | GSK2578215A |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5361 |
| Prices | $225.00, $925.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 1285515-21-0 |
| Chemical Name | 5-(2-Fluoro-4-pyridinyl)-2-(phenylmethoxy)-N-3-pyridinylbenzamide |
| Formula | C24H18FN3O2 |
| Molecular Weight | 399.42 |
| Purity | >99 % |
| Description | Potent LRRK2 inhibitor (IC 50 values are 8.9 and 10.1 nM for LRRK2[G2019S] mutant and wild-type LRRK2 respectively). Displays selectivity for LRRK2 over a panel of 460 other kinases. Blocks Ser910 and Ser935 phosphorylation in vitro and in peripheral tissues in vivo . Brain penetrant. |
| Supplier Page | Shop |