| Name | GW 803430 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 3385 |
| Prices | $225.00, $925.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 515141-51-2 |
| Chemical Name | 6-(4-Chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3H)-one |
| Formula | C25H24ClN3O3S |
| Molecular Weight | 481.99 |
| Purity | >99 % |
| Description | Selective melanin-concentrating hormone receptor 1 (MCH 1 ) antagonist (IC 50 = 9.3 nM). Displays antiobesity and antidepressant-like effects in rats and mice. Orally active. |
| Supplier Page | Shop |
Rivera G, Bocanegra-Garcia V, Galiano S, Cirauqui N, Ceras J, Perez S, Aldana I, Monge A. Curr Med Chem. 2008;15(10):1025-43.
Gehlert DR, Rasmussen K, Shaw J, Li X, Ardayfio P, Craft L, Coskun T, Zhang HY, Chen Y, Witkin JM. J Pharmacol Exp Ther. 2009 May;329(2):429-38.