Name | H2L5186303 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 4870 |
Prices | $189.00, $765.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 139262-76-3 |
Chemical Name | (Z,Z)-4,4'-[1,3-Phenylenebis(oxy-4,1-phenyleneimino)]bis[4-oxo-2-butenoicacid |
Formula | C26H20N2O8 |
Molecular Weight | 488.45 |
Purity | >98 % |
Description | Potent and selective lysophosphatidic acid 2 (LPA 2 ) receptor antagonist (IC 50 values are 8.9, 1230 and 27354 nM for LPA 2 , LPA 3 and LPA 1 receptors respectively, in a LPA-elicited calcium mobilization assay). |
Supplier Page | Shop |
Fells JI, Tsukahara R, Fujiwara Y, Liu J, Perygin DH, Osborne DA, Tigyi G, Parrill AL. Bioorg Med Chem. 2008 Jun 1;16(11):6207-17.
Fells JI, Tsukahara R, Liu J, Tigyi G, Parrill AL. Bioorg Med Chem. 2009 Nov 1;17(21):7457-64.