Harmine

Name Harmine
Supplier Tocris Bioscience
Catalog 1132
Prices $59.00
Sizes 50 mg
Function Type Inhibitor
Cas Number 442-51-3
Chemical Name 7-Methoxy-1-methyl-9H-pyrido[3,4-b]indole
Formula C13H12N2O
Molecular Weight 212.25
Purity >98 %
Description Potent and selective inhibitor of DYRK1A (IC 50 values are 80, 800 and 900 nM for DYRK1A, DYRK3 and DYRK2 respectively). Inhibits DYRK1A-mediated tau phosphorylation and regulates PPAR γ expression. Also induces pancreatic beta cell proliferation. Exhibits antidiabetic activity. Orally bioavailable.
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Product References

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The small molecule harmine is an antidiabetic cell-type-specific regulator of - The small molecule harmine is an antidiabetic cell-type-specific regulator of

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