8-Hydroxy-DPAT hydrobromide

Name 8-Hydroxy-DPAT hydrobromide
Supplier Tocris Bioscience
Catalog 0706
Prices $69.00, $255.00
Sizes 10 mg, 50 mg
Function Type Agonist
Cas Number 76135-31-4
Chemical Name (±)-8-Hydroxy-2-dipropylaminotetralinhydrobromide
Formula C16H25NO.HBr
Molecular Weight 328.29
Purity >98 %
Description The standard selective 5-HT 1A agonist. Also has moderate affinity for 5-HT 7 receptors (pK i is 6.6 at the human 5-HT 7 receptor expressed in HEK 293 cells). Reduces hippocampal 5-HT levels following systemic administration in rats in vivo . ( R )-(+)-8-Hydroxy-DPAT hydrobromide (Cat. No. 1080) and 7-Hydroxy-DPAT hydrobromide (Cat. No. 0706) also available.
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Product References

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Antagonist activity of meta-chlorophenylpiperazine and partial agonist activity - Antagonist activity of meta-chlorophenylpiperazine and partial agonist activity

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