| Name | I-CBP 112 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5066 |
| Prices | $255.00, $1,045.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Chemical Name | 1-[7-(3,4-Dimethoxyphenyl)-9-[[(3S)-1-methylpiperidin-3-yl]methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one |
| Formula | C27H36N2O5 |
| Molecular Weight | 468.59 |
| Purity | >98 % |
| Description | CBP/p300 bromodomain inhibitor (IC 50 values are 0.142-0.17 and 0.625 μ M for CBP and p300 respectively). Selective for CBP and p300 over ATAD2, BAZ2B, BRD2(2), BRD4(1), PB1(5), PCAF, PHIP(2) and TIF1 α bromodomains in a BLI assay. Accelerates FRAP recovery in cells at a concentration of 1 μ M. |
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