Immepip dihydrobromide

• Supplier: Tocris Bioscience
• Catalog: 3700
• Prices: $159.00, $665.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 164391-47-3
• Chemical Name: 4-(1H-Imidazol-4-ylmethyl)piperidinedihydrobromide
• Formula: C9H15N3.2HBr
• Molecular Weight: 327.06
• Description: Potent histamine H 3 receptor agonist. Also binds to H 4 receptors (K i values are 0.4 and 9 nM at human recombinant H 3 and H 4 receptors respectively). Equipotent to or slightly more active than (R)- α -methylhistamine at H 3 receptors.

Product References

A new potent and selective histamine H3 receptor agonist, - A new potent and selective histamine H3 receptor agonist,

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Cardiovascular effects of selective agonists and antagonists of histamine H3 - Cardiovascular effects of selective agonists and antagonists of histamine H3

Coruzzi G, Gambarelli E, Bertaccini G, Timmerman H. Naunyn Schmiedebergs Arch Pharmacol. 1995 Jun;351(6):569-75.

Cloning and pharmacological characterization of a fourth histamine receptor - Cloning and pharmacological characterization of a fourth histamine receptor

Liu C, Ma X, Jiang X, Wilson SJ, Hofstra CL, Blevitt J, Pyati J, Li X, Chai W, Carruthers N, Lovenberg TW. Mol Pharmacol. 2001 Mar;59(3):420-6.