5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative

• Supplier: Tocris Bioscience
• Catalog: 1518
• Prices: $129.00
• Sizes: 200 µg
• Cas Number: 213766-21-3
• Chemical Name: (2S)-2-[[[5-(Trimethylstannyl)-3-pyridinyl]oxy]methyl]-1-azetidinecarboxylicacid,t-butylester
• Formula: C17H28N2O3Sn
• Molecular Weight: 427.11
• Purity: >98 %
• Description: Precursor to the highly potent and selective ligand for the α 4 β 2 nicotinic receptor, 5-Iodo-A-85380 (Cat. No.1518). Suitable for radioiodination.

Product References

2-, 5-, and 6-Halo-3-(2(S)-azetidinylmethoxy)pyridines: synthesis, affinity for - 2-, 5-, and 6-Halo-3-(2(S)-azetidinylmethoxy)pyridines: synthesis, affinity for

Koren AO, Horti AG, Mukhin AG, Gundisch D, Kimes AS, Dannals RF, London ED. J Med Chem. 1998 Sep 10;41(19):3690-8.

5-Iodo-A-85380, an alpha4beta2 subtype-selective ligand for nicotinic - 5-Iodo-A-85380, an alpha4beta2 subtype-selective ligand for nicotinic

Mukhin AG, Gundisch D, Horti AG, Koren AO, Tamagnan G, Kimes AS, Chambers J, Vaupel DB, King SL, Picciotto MR, Innis RB, London ED. Mol Pharmacol. 2000 Mar;57(3):642-9.