Name | 5'-Iodoresiniferatoxin |
---|---|
Supplier | Tocris Bioscience |
Catalog | 0779 |
Prices | $369.00 |
Sizes | 1 mg |
Function Type | Antagonist |
Cas Number | 535974-91-5 |
Chemical Name | 6,7-Deepoxy-6,7-didehydro-5-deoxy-21-dephenyl-21-(phenylmethyl)-daphnetoxin,20-(4-hydroxy-5-iodo-3-methoxybenzeneacetate) |
Formula | C37H39IO9 |
Molecular Weight | 754.6 |
Purity | >98 % |
Description | Potent and silent vanilloid receptor antagonist, 40-fold more potent than capsazepine (Cat. No. 0464). Binds to TRPV1 (VR1) receptors expressed in HEK293 cells with a K i of 5.8 nM. |
Supplier Page | Shop |
Wahl P, Foged C, Tullin S, Thomsen C. Mol Pharmacol. 2001 Jan;59(1):9-15.
Marinelli S, Vaughan CW, Christie MJ, Connor M. J Physiol. 2002 Sep 1;543(Pt 2):531-40.