JNJ DGAT2-A

Name JNJ DGAT2-A
Supplier Tocris Bioscience
Catalog 4021
Prices $299.00
Sizes 10 mg
Function Type Inhibitor
Cas Number 1962931-71-0
Chemical Name 3-Bromo-4-[2-fluoro-4-[[4-oxo-2-[[2-(pyridin-2-yl)ethyl]amino]-1,3-thiazol-5-(4H)ylidene]methyl]phenoxy]benzonitrile
Formula C24H16BrFN4O2S
Molecular Weight 523.38
Description DGAT2 inhibitor (IC 50 = 140 nM). Exhibits >70-fold selectivity for DGAT2 over DGAT1 and MGAT2.
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Product References

Pharmacological characterization and CNS effects of a novel highly selective - Pharmacological characterization and CNS effects of a novel highly selective

Sallinen J, Hoglund I, Engstrom M, Lehtimaki J, Virtanen R, Sirvio J, Wurster S, Savola JM, Haapalinna A. Br J Pharmacol. 2007 Feb;150(4):391-402. Epub 2007 Jan 15.

JP-1302: a new tool to shed light on the roles of alpha2C-adrenoceptors in brain. - JP-1302: a new tool to shed light on the roles of alpha2C-adrenoceptors in brain.

Tricklebank MD. Br J Pharmacol. 2007 Feb;150(4):381-2. Epub 2007 Jan 15.