JTE 907

• Supplier: Tocris Bioscience
• Catalog: 5185
• Prices: $199.00, $825.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 282089-49-0
• Chemical Name: N-(1,3-Benzodioxol-5-ylmethyl)-1,2-dihydro-7-methoxy-2-oxo-8-(pentyloxy)-3-quinolinecarboxamide
• Formula: C24H26N2O6
• Molecular Weight: 438.48
• Purity: >99 %
• Description: Highly selective cannabinoid CB 2 receptor inverse agonist. Binds with high affinity to rat, mouse and human CB 2 receptors (K i values are 0.38, 1.55 and 35.9 nM respectively). Produces anti-inflammatory effects in vivo .

Product References

In vitro and in vivo pharmacological characterization of JTE-907, a novel - In vitro and in vivo pharmacological characterization of JTE-907, a novel

Iwamura H, Suzuki H, Ueda Y, Kaya T, Inaba T. J Pharmacol Exp Ther. 2001 Feb;296(2):420-5.

Involvement of cannabinoid CB(2) receptor-mediated response and efficacy of - Involvement of cannabinoid CB(2) receptor-mediated response and efficacy of

Ueda Y, Miyagawa N, Matsui T, Kaya T, Iwamura H. Eur J Pharmacol. 2005 Sep 27;520(1-3):164-71.

The cannabinoid CB2 receptor inverse agonist JTE-907 suppresses spontaneous - The cannabinoid CB2 receptor inverse agonist JTE-907 suppresses spontaneous

Maekawa T, Nojima H, Kuraishi Y, Aisaka K. Eur J Pharmacol. 2006 Aug 7;542(1-3):179-83. Epub 2006 Jun 2.