| Name | KB SRC 4 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 3962 |
| Prices | $255.00, $1,045.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 1380088-03-8 |
| Chemical Name | 1-[3-[1-([1,1'-Biphenyl]-3-ylmethyl)-1H-1,2,3-triazol-5-yl]phenyl]-3-(4-chlorophenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |
| Formula | C32H23ClN8 |
| Molecular Weight | 555.03 |
| Purity | >98 % |
| Description | Potent and selective c-Src inhibitor (K i = 44 nM); does not inhibit c-Abl at concentrations up to 125 μ M. Selective between Src family members (K d values are 86, 160, 240, 720, 3200, 4400, and >40,000 nM for c-Src, Lck, Fgr, Yes, Lyn, Hck and Fyn respectively). Significantly inhibits cell growth in 4T1 mammary carcinoma tumor cells. |
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