| Name | L-651,582 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2410 |
| Prices | $199.00, $825.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Blocker |
| Cas Number | 99519-84-3 |
| Chemical Name | 5-Amino-1-[[3,5-dichloro-4-(4-chlorobenzoyl)phenyl]methyl]-1H-1,2,3-triazole-4-carboxamide |
| Formula | C17H12Cl3N5O2 |
| Molecular Weight | 424.67 |
| Purity | >98 % |
| Description | Orally active Ca 2+ channel blocker; inhibits K + - and carbachol-stimulated Ca 2+ influx (IC 50 values are 500 and 935 nM respectively). Exhibits antiproliferative, antiangiogenic and antimetastatic activity in vivo and displays selectivity towards numerous mismatch repair-deficient tumor cell lines in vitro . |
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