L-694,247

• Supplier: Tocris Bioscience
• Catalog: 0426
• Prices: $195.00, $805.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 137403-12-4
• Chemical Name: 2-[5-[3-(4-Methylsulfonylamino)benzyl-1,2,4-oxadiazol-5-yl]-1H-indol-3-yl]ethanamine
• Formula: C20H21N5O3S
• Molecular Weight: 411.48
• Purity: >98 %
• Description: Selective and extremely potent 5-HT 1D receptor agonist.

Product References

L-694,247: a potent 5-HT1D receptor agonist. - L-694,247: a potent 5-HT1D receptor agonist.

Beer MS, Stanton JA, Bevan Y, Heald A, Reeve AJ, Street LJ, Matassa VG, Hargreaves RJ, Middlemiss DN. Br J Pharmacol. 1993 Nov;110(3):1196-200.

Synthesis and serotonergic activity of 5-(oxadiazolyl)tryptamines: potent - Synthesis and serotonergic activity of 5-(oxadiazolyl)tryptamines: potent

Street LJ, Baker R, Castro JL, Chambers MS, Guiblin AR, Hobbs SC, Matassa VG, Reeve AJ, Beer MS, Middlemiss DN, et al.. J Med Chem. 1993 May 28;36(11):1529-38.

[3H]L-694,247 labels the 5-HT1D beta receptor in pig caudate membranes. - [3H]L-694,247 labels the 5-HT1D beta receptor in pig caudate membranes.

Heald A, Stanton JA, Osborne SA, Middlemiss DN, Beer MS. Eur J Pharmacol. 1994 Oct 24;264(2):213-6.

Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in - Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in

Buhlen M, Fink K, Boing C, Gothert M. Naunyn Schmiedebergs Arch Pharmacol. 1996 Feb;353(3):281-9.