Name | L-759,656 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 2197 |
Prices | $255.00 |
Sizes | 10 mg |
Function Type | Agonist |
Cas Number | 174627-56-6 |
Chemical Name | (6aR,10aR)-3-(1,1-Dimethylheptyl)-6a,7,8,9,10,10a-hexahydro-1-methoxy-6,6-dimethyl-9-methylene-6H-dibenzo[b,d]pyran |
Formula | C26H40O2 |
Molecular Weight | 384.6 |
Purity | >98 % |
Description | Highly selective CB 2 receptor agonist (K i values are 11.8 and 4888 nM for CB 2 and CB 1 receptors respectively). Potently inhibits forskolin-stimulated cAMP production via CB 2 receptors expressed in CHO cells (EC 50 = 3.1 nM). |
Supplier Page | Shop |
Ross RA, Brockie HC, Stevenson LA, Murphy VL, Templeton F, Makriyannis A, Pertwee RG. Br J Pharmacol. 1999 Feb;126(3):665-72.
Huffman JW. Mini Rev Med Chem. 2005 Jul;5(7):641-9.