L-759,633

Name L-759,633
Supplier Tocris Bioscience
Catalog 2434
Prices $255.00
Sizes 10 mg
Function Type Agonist
Cas Number 174627-50-0
Chemical Name (6aR,10aR)-3-(1,1-Dimethylheptyl)-6a,7,10,10a-tetrahydro-1-methoxy-6,6,9-trimethyl-6H-dibenzo[b,d]pyran
Formula C26H40O2
Molecular Weight 384.59
Purity >98 %
Description High affinity, selective CB 2 receptor agonist (K i values are 6.4 and 1043 nM for CB 2 and CB 1 receptors respectively). Potently inhibits forskolin-stimulated cAMP production via CB 2 receptors expressed in CHO cells (EC 50 = 8.1 nM).
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Product References

3-(1',1'-Dimethylbutyl)-1-deoxy-delta8-THC and related compounds: synthesis of - 3-(1',1'-Dimethylbutyl)-1-deoxy-delta8-THC and related compounds: synthesis of

Huffman JW, Liddle J, Yu S, Aung MM, Abood ME, Wiley JL, Martin BR. Bioorg Med Chem. 1999 Dec;7(12):2905-14.

Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of - Agonist-inverse agonist characterization at CB1 and CB2 cannabinoid receptors of

Ross RA, Brockie HC, Stevenson LA, Murphy VL, Templeton F, Makriyannis A, Pertwee RG. Br J Pharmacol. 1999 Feb;126(3):665-72.