L-803,087 trifluoroacetate

Name	L-803,087 trifluoroacetate
Supplier	Tocris Bioscience
Catalog	2235
Prices	$279.00
Sizes	10 mg
Function Type	Agonist
Cas Number	217480-26-7
Chemical Name	N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-argininemethylestertrifluoroacetate
Formula	C25H29F2N5O3.CF3CO2H
Molecular Weight	599.56
Purity	>97 %
Description	Potent and selective somatostatin sst 4 receptor agonist. K i values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst 4 , sst 1 , sst 2 , sst 3 and sst 5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo .
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Product References

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Identification and characterization of subtype selective somatostatin receptor - Identification and characterization of subtype selective somatostatin receptor

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Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and - Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and

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