| Name | L-817,818 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 1979 |
| Prices | $279.00 |
| Sizes | 10 mg |
| Function Type | Agonist |
| Cas Number | 217480-27-8 |
| Chemical Name | N2-[[2-(2-Naphthalenyl)-1H-benz[g]indol-3-yl]acetyl-D-lysine(2S)-2-aminopropylester |
| Formula | C33H36N4O3 |
| Molecular Weight | 536.67 |
| Purity | >99 % |
| Description | Potent and selective somatostatin sst 5 receptor agonist. K i values are 0.4, 3.3, 52, 64 and 82 nM for cloned human sst 5 , sst 1 , sst 2 , sst 3 and sst 4 receptors respectively. Inhibits growth hormone release from rat pituitary cells (EC 50 = 3.1 nM) and insulin release from mouse pancreatic islets (EC 50 = 0.3 nM) in vitro . |
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Chen G, Bower KA, Ma C, Fang S, Thiele CJ, Luo J. FASEB J. 2004 Jul;18(10):1162-4. Epub 2004 May 7.
Kaidanovich-Beilin O, Milman A, Weizman A, Pick CG, Eldar-Finkelman H. Biol Psychiatry. 2004 Apr 15;55(8):781-4.