LY 288513

• Supplier: Tocris Bioscience
• Catalog: 3077
• Prices: $279.00, $1,145.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 147523-65-7
• Chemical Name: (4S,5R)-N-(4-Bromophenyl)-3-oxo-4,5-diphenyl-1-pyrazolidinecarboxamide
• Formula: C22H18BrN3O2
• Molecular Weight: 436.3
• Purity: >98 %
• Description: Selective CCK 2 receptor antagonist (IC 50 values are 16 and > 30,000 nM for CCK 2 and CCK 1 respectively). Displays anxiolytic and antipsychotic properties in vivo .

Product References

CCK, schizophrenia, and anxiety. CCK-B antagonists inhibit the activity of brain - CCK, schizophrenia, and anxiety. CCK-B antagonists inhibit the activity of brain

Rasmussen K. Ann N Y Acad Sci. 1994 Mar 23;713:300-11.

Central nervous system characterization of the new cholecystokininB antagonist - Central nervous system characterization of the new cholecystokininB antagonist

Helton DR, Berger JE, Czachura JF, Rasmussen K, Kallman MJ. Pharmacol Biochem Behav. 1996 Mar;53(3):493-502.