| Name | MA 2029 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2698 |
| Prices | $209.00, $879.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 287206-61-5 |
| Chemical Name | 4-Fluoro-N-methyl-L-phenylalanyl-N-methyl-L-valyl-3-(1,1-dimethylethyl)-N-ethyl-L-tyrosinamide |
| Formula | C31H45FN4O4 |
| Molecular Weight | 556.71 |
| Purity | >98 % |
| Description | Potent and selective, competitive motilin receptor antagonist (IC 50 = 4.9 nM). Selective for the motilin receptor over a range of other receptors and ion channels. Inhibits motilin-induced duodenal muscle contractions in vitro . Also inhibits motilin-induced colonic and abdominal contractions in vivo . Orally active. |
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