Name | MDA 19 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 0337 |
Prices | $175.00, $709.00 |
Sizes | 10 mg, 50 mg |
Function Type | Agonist |
Cas Number | 1048973-47-2 |
Chemical Name | N'-[(3Z)-1-Hexyl-2-oxo-1,2-dihydro-3H-indol-3-ylidene]benzohydrazide |
Formula | C21H23N3O2 |
Molecular Weight | 349.43 |
Purity | >99 % |
Description | CB 2 receptor agonist. Displays 4-fold higher affinity for the human CB 2 receptor than the human CB 1 receptor (K i values are 43.3 and 162.4 nM respectively); shows 70-fold affinity for the rat CB 2 receptor over the rat CB 1 receptor (K i values are 16.3 and 1130 nM respectively). Attenuates tactile allodynia in a rat model; does not affect rat locomotor activity. |
Supplier Page | Shop |
Diaz P, Xu J, Astruc-Diaz F, Pan HM, Brown DL, Naguib M. J Med Chem. 2008 Aug 28;51(16):4932-47.
Xu JJ, Diaz P, Astruc-Diaz F, Craig S, Munoz E, Naguib M. Anesth Analg. 2010 Jul;111(1):99-109.