Metergoline

• Supplier: Tocris Bioscience
• Catalog: 1443
• Prices: $69.00, $255.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 17692-51-2
• Chemical Name: [(8β)-1,6-Dimethylergolin-8-yl)methyl]carbamicacidphenylmethylester
• Formula: C25H29N3O2
• Molecular Weight: 403.52
• Description: Antagonist at 5-HT 1 /5-HT 2 with activity at 5-HT 1D . Has moderate affinity for 5-HT 6 and high affinity for 5-HT 7 .

Product References

Effects of various serotonin receptor subtype-selective antagonists alone and on - Effects of various serotonin receptor subtype-selective antagonists alone and on

Aulakh CS, Hill JL, Murphy DL. J Pharmacol Exp Ther. 1992 Nov;263(2):588-95.

Pharmacological characterization of serotonin receptor subtypes involved in - Pharmacological characterization of serotonin receptor subtypes involved in

Bagdy G, Sved AF, Murphy DL, Szemeredi K. Eur J Pharmacol. 1992 Jan 21;210(3):285-9.

Agonist activity of sumatriptan and metergoline at the human 5-HT1D beta - Agonist activity of sumatriptan and metergoline at the human 5-HT1D beta

Miller KJ, King A, Demchyshyn L, Niznik H, Teitler M. Eur J Pharmacol. 1992 Sep 1;227(1):99-102.