Name | ( R )-MG 132 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 1748 |
Prices | $275.00 |
Sizes | 10 mg |
Function Type | Inhibitor |
Cas Number | 1211877-36-9 |
Chemical Name | N-[(Phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-D-leucinamide |
Formula | C26H41N3O5 |
Molecular Weight | 475.63 |
Purity | >98 % |
Description | Potent 20S proteasome inhibitor (IC 50 = 0.22 nM). Exhibits cytostatic and cytotoxic effects in tumor cells in vitro . |
Supplier Page | Shop |
Gotti C, Balestra B, Moretti M, Rovati GE, Maggi L, Rossoni G, Berti F, Villa L, Pallavicini M, Clementi F. Br J Pharmacol. 1998 Jul;124(6):1197-206.
Maggi L, Palma E, Eusebi F, Moretti M, Balestra B, Clementi F, Gotti C. Br J Pharmacol. 1999 Jan;126(1):285-95.