MRS 2211

Name MRS 2211
Supplier Tocris Bioscience
Catalog 0900
Prices $109.00, $459.00
Sizes 10 mg, 50 mg
Function Type Antagonist
Chemical Name 2-[(2-Chloro-5-nitrophenyl)azo]-5-hydroxy-6-methyl-3-[(phosphonooxy)methyl]-4-pyridinecarboxaldehydedisodiumsalt
Formula C14H10N4O8Na2PCl
Molecular Weight 474.66
Purity >96 %
Description Competitive P2Y 13 receptor antagonist (pIC 50 = 5.97) that displays > 20-fold selectivity over P2Y 1 and P2Y 12 receptors.
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Product References

Synthesis of pyridoxal phosphate derivatives with antagonist activity at the - Synthesis of pyridoxal phosphate derivatives with antagonist activity at the

Kim YC, Lee JS, Sak K, Marteau F, Mamedova L, Boeynaems JM, Jacobson KA. Biochem Pharmacol. 2005 Jul 15;70(2):266-74.

Pharmacological profiles of cloned mammalian P2Y-receptor subtypes. - Pharmacological profiles of cloned mammalian P2Y-receptor subtypes.

von Kugelgen I. Pharmacol Ther. 2006 Jun;110(3):415-32. Epub 2005 Oct 28.