Naloxone 3-glucuronide carbonic acid salt

Name Naloxone 3-glucuronide carbonic acid salt
Supplier Tocris Bioscience
Catalog 0599
Prices $99.00
Sizes 1 mg
Chemical Name (5α)-4,5-Epoxy-14-hydroxy-6-oxo-17-(2-propenyl)morphinan-3-ylβ-D-glucopyranosiduronicacidcarbonicacidsalt
Formula C25H29NO10.H2CO3
Molecular Weight 565.52
Purity >98 %
Description Naloxone conjugate. Following oral administration induces delayed diarrhea, as well as milder and delayed withdrawal behavior and tail skin temperature (TST) response compared with naloxone in morphine-dependent rats.
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Product References

Pharmacological actions of a novel mixed opiate agonist/antagonist: naloxone - Pharmacological actions of a novel mixed opiate agonist/antagonist: naloxone

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Has the sun set on kappa3-opioid receptors? - Has the sun set on kappa3-opioid receptors?

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Agonist activity of naloxone benzoylhydrazone at recombinant and native opioid - Agonist activity of naloxone benzoylhydrazone at recombinant and native opioid

Olianas MC, Concas D, Onali P. Br J Pharmacol. 2006 Feb;147(4):360-70.