Naltriben mesylate

• Supplier: Tocris Bioscience
• Catalog: 0677
• Prices: $155.00, $645.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 122517-78-6
• Chemical Name: 17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate
• Formula: C26H25NO4.CH3SO3H
• Molecular Weight: 511.59
• Description: Selective and potent δ -opioid receptor antagonist (K i values are 0.013, 19 and 152 nM for δ , μ and κ receptors respectively). Displays selectivity for the δ 2 subtype in vivo .

Product References

Role of spacer and address components in peptidomimetic delta opioid receptor - Role of spacer and address components in peptidomimetic delta opioid receptor

Portoghese PS, Nagase H, MaloneyHuss KE, Lin CE, Takemori AE. J Med Chem. 1991 May;34(5):1715-20.

Involvement of delta 2 opioid receptors in the development of morphine dependence - Involvement of delta 2 opioid receptors in the development of morphine dependence

Miyamoto Y, Portoghese PS, Takemori AE. J Pharmacol Exp Ther. 1993 Mar;264(3):1141-5.

Modulation of nociception by microinjection of delta-1 and delta-2 opioid - Modulation of nociception by microinjection of delta-1 and delta-2 opioid

Thorat SN, Hammond DL. J Pharmacol Exp Ther. 1997 Dec;283(3):1185-92.