Naltrindole hydrochloride

• Supplier: Tocris Bioscience
• Catalog: 0892
• Prices: $139.00, $575.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 111469-81-9
• Chemical Name: 17-(Cyclopropylmethyl)-6,7-dehydro-4,5α-epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinanhydrochloride
• Formula: C26H26N2O3.HCl
• Molecular Weight: 450.96
• Purity: >99 %
• Description: Highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ and κ opioid receptors.

Product References

Design of peptidomimetic delta opioid receptor antagonists using the - Design of peptidomimetic delta opioid receptor antagonists using the

Portoghese PS, Sultana M, Takemori AE. J Med Chem. 1990 Jun;33(6):1714-20.

Naltrindole, an opioid delta antagonist, blocks the enhancement of - Naltrindole, an opioid delta antagonist, blocks the enhancement of

Ossipov MH, Kovelowski CJ, Vanderah T, Porreca F. Neurosci Lett. 1994 Nov 7;181(1-2):9-12.

The delta-opioid receptor antagonist naltrindole prevents sensitization to the - The delta-opioid receptor antagonist naltrindole prevents sensitization to the

Shippenberg TS, Heidbreder C. Eur J Pharmacol. 1995 Jun 23;280(1):55-61.