NCT 501 hydrochloride

• Supplier: Tocris Bioscience
• Catalog: 0780
• Prices: $259.00, $1,089.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Chemical Name: 8-[[4-(Cyclopropylcarbonyl)-1-piperazinyl]methyl]-3,7-dihydro-1,3-dimethyl-7-(3-methylbutyl)-1H-purine-2,6-dionehydrochloride
• Formula: C21H32N6O3.HCl
• Molecular Weight: 452.98
• Purity: >98 %
• Description: Potent and selective ALDH1A1 inhibitor (IC 50 = 40 nM). Exhibits >1000-fold selectivity for ALDH1A1 over ALDH3A1, ALDH1B1, ALDH2, HPGD and HSD17 β 4. Also selective over a panel of 168 GPCRs. Blood-brain barrier permeable.

Product References

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