NF 449

• Supplier: Tocris Bioscience
• Catalog: 3830
• Prices: $205.00, $845.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 627034-85-9
• Chemical Name: 4,4',4'',4'''-[Carbonylbis(imino-5,1,3-benzenetriyl-bis(carbonylimino))]tetrakis-1,3-benzenedisulfonicacid,octasodiumsalt
• Formula: C41H24N6Na8O29S8
• Molecular Weight: 1505.06
• Description: Potent purinergic receptor antagonist that displays high selectivity for P2X 1 (IC 50 values are 0.28, 0.69, 120, 1820, 47000 and > 300000 nM for rP2X 1 , rP2X 1+5 , rP2X 2+3 , rP2X 3 , rP2X 2 and P2X 4 receptors respectively). Provides antithrombotic protection in vivo . Also acts as a G s α -selective antagonist.

Product References

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