| Name | NI 42 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5363 |
| Prices | $179.00, $745.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 1884640-99-6 |
| Chemical Name | 4-Cyano-N-(1,2-dihydro-1,3-dimethyl-2-oxo-6-quinolinyl)benzenesulfonamide |
| Formula | C18H15N3O3S |
| Molecular Weight | 353.39 |
| Purity | >98 % |
| Description | High affinity BRPF inhibitor (K d values are 40, 210 and 943 nM for BRPF1B, 2 and 3, respectively). Also exhibits modest activity at BRD9 (K d = 1130 nM). Exhibits selectivity for BRPF over 44 other bromodomains. Orally bioavailable. |
| Supplier Page | Shop |