Name | NIDA 41020 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3546 |
Prices | $189.00, $765.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 502486-89-7 |
Chemical Name | N-(Piperidin-1-yl)-5-(4-methoxyphenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide |
Formula | C23H24Cl2N4O2 |
Molecular Weight | 459.37 |
Purity | >99 % |
Description | High affinity CB 1 receptor antagonist (K i = 4.1 nM). Exhibits significantly reduced lipophilicity compared to other CB 1 antagonists. |
Supplier Page | Shop |
Katoch-Rouse R, Pavlova OA, Caulder T, Hoffman AF, Mukhin AG, Horti AG. J Med Chem. 2003 Feb 13;46(4):642-5.
Miller DK, Rodvelt KR, Constales C, Putnam WC. Life Sci. 2007 Jun 13;81(1):63-71. Epub 2007 May 1.