[Lys 5 ,MeLeu 9 ,Nle 10 ]-NKA(4-10)

• Supplier: Tocris Bioscience
• Catalog: 5293
• Prices: $199.00
• Sizes: 1 mg
• Function Type: Agonist
• Cas Number: 137565-28-7
• Formula: C39H65N9O9
• Molecular Weight: 804
• Description: Highy selective and potent NK 2 receptor agonist (IC 50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC 50 values are 117 and 10 nM respectively).

Product References

Selective agonists of NK-2 binding sites highly active on rat portal vein (NK-3 - Selective agonists of NK-2 binding sites highly active on rat portal vein (NK-3

Chassaing G, Lavielle S, Loeuillet D, Robilliard P, Carruette A, Garret C, Beaujouan JC, Saffroy M, Petitet F, Torrens Y, et al.. Neuropeptides. 1991 Jun;19(2):91-5.

An investigation of tachykinin NK2 receptor subtypes in the rat. - An investigation of tachykinin NK2 receptor subtypes in the rat.

Matuszek MA, Zeng XP, Strigas J, Burcher E. Eur J Pharmacol. 1998 Jul 3;352(1):103-9.

Tachykinin NK2 receptor and functional mechanisms in human colon: changes with - Tachykinin NK2 receptor and functional mechanisms in human colon: changes with

Burcher E, Shang F, Warner FJ, Du Q, Lubowski DZ, King DW, Liu L. J Pharmacol Exp Ther. 2008 Jan;324(1):170-8. Epub 2007 Oct 24.