| Name | NNC 55-0396 dihydrochloride |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2440 |
| Prices | $259.00 |
| Sizes | 10 mg |
| Function Type | Blocker |
| Cas Number | 357400-13-6 |
| Chemical Name | (1S,2S)-2-[2-[[3-(1H-Benzimidazol-2-yl)propyl]methylamino]ethyl]-6-fluoro-1,2,3,4-tetrahydro-1-(1-methylethyl)-2-naphthalenylcyclopropanecarboxylatedihydrochloride |
| Formula | C30H38FN3O2.2HCl |
| Molecular Weight | 564.57 |
| Purity | >98 % |
| Description | Highly selective T-type calcium channel blocker. Displays IC 50 values of 6.8 and > 100 μ M for inhibition of Ca v 3.1 T-type channels and HVA currents respectively in INS-1 cells. |
| Supplier Page | Shop |
Huang L, Keyser BM, Tagmose TM, Hansen JB, Taylor JT, Zhuang H, Zhang M, Ragsdale DS, Li M. J Pharmacol Exp Ther. 2004 Apr;309(1):193-9. Epub 2004 Jan 12.
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