| Name | NS 3861 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2187 |
| Prices | $139.00, $585.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Agonist |
| Cas Number | 216853-60-0 |
| Chemical Name | 3-(3-Bromo-2-thienyl)-8-methyl-8-azabicyclo[3.2.1]oct-2-enefumarate |
| Formula | C12H14BrNS.C4H4O4 |
| Molecular Weight | 400.29 |
| Purity | >98 % |
| Description | α 3 β 2 full agonist (EC 50 = 1.6 μ M). Also α 3 β 4 partial agonist (EC 50 = 1 μ M). Exhibits minimal activity at α 4 β 2 and α 4 β 4. Displays high affinity for α 3 β 4, α 4 β 4, α 3 β 2 and α 4 β 2 (K i values are 0.62, 7.8, 25 and 55 nM respectively). |
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