Octreotide

• Supplier: Tocris Bioscience
• Catalog: 2242
• Prices: $259.00
• Sizes: 1 mg
• Function Type: Agonist
• Cas Number: 83150-76-9
• Formula: C49H66N10O10S2
• Molecular Weight: 1019.24
• Description: Peptide agonist for sst 2 , sst 3 and sst 5 somatostatin receptors. IC 50 /K d values (nM) at cloned human somatostatin receptors are: 290 - 1140 (sst 1 ), 0.4 - 2.1 (sst 2 ), 4.4 - 34.5 (sst 3 ), > 1000 (sst 4 ), and 5.6 - 32 (sst 5 ).

Product References

Cloned somatostatin receptors: identification of subtype-selective peptides and - Cloned somatostatin receptors: identification of subtype-selective peptides and

Raynor K, Murphy WA, Coy DH, Taylor JE, Moreau JP, Yasuda K, Bell GI, Reisine T. Mol Pharmacol. 1993 Jun;43(6):838-44.

Molecular pharmacology of somatostatin receptors. - Molecular pharmacology of somatostatin receptors.

Hoyer D, Lubbert H, Bruns C. Naunyn Schmiedebergs Arch Pharmacol. 1994 Nov;350(5):441-53.