Name | OLDA |
---|---|
Supplier | Tocris Bioscience |
Catalog | 5542 |
Prices | $109.00, $455.00 |
Sizes | 5 mg, 25 mg |
Function Type | Agonist |
Cas Number | 105955-11-1 |
Chemical Name | (9Z)-N-[2-(3,4-Dihydroxyphenyl)ethyl]-9-octadecenamide |
Formula | C26H43NO3 |
Molecular Weight | 417.63 |
Purity | >99 % |
Description | Potent endogenous vanilloid TRPV1 (VR1) receptor agonist (EC 50 = 36 nM at hVR1) with low affinity for rCB 1 receptors (K i = 1.6 μ M). Potently induces VR1-mediated thermal hyperalgesia in rats in vivo . |
Supplier Page | Shop |
Chu CJ, Huang SM, De Petrocellis L, Bisogno T, Ewing SA, Miller JD, Zipkin RE, Daddario N, Appendino G, Di Marzo V, Walker JM. J Biol Chem. 2003 Apr 18;278(16):13633-9. Epub 2003 Feb 4.
Butelman ER, Harris TJ, Kreek MJ. J Pharmacol Exp Ther. 2004 Oct;311(1):155-63. Epub 2004 May 19.