Oleanolic acid

• Supplier: Tocris Bioscience
• Catalog: 0878
• Prices: $65.00
• Sizes: 50 mg
• Function Type: Agonist
• Cas Number: 508-02-1
• Chemical Name: (3β)-3-Hydroxyolean-12-en-28-oicacid
• Formula: C30H48O3
• Molecular Weight: 456.7
• Purity: >97 %
• Description: GPBA receptor (TGR5) partial agonist (EC 50 = 2.25 μ M; 72% efficacy). Displays no activity at FXR. Also inhibits protein phosphate 1B (PTP1B) and glycogen phosphorylase. Suppresses cell proliferation and increases apoptosis in T24 bladder cancer cells. Antidiabetic, antihyperglycaemic, antitumor and hepatoprotective.

Product References

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