Oleylethanolamide

• Supplier: Tocris Bioscience
• Catalog: 3854
• Prices: $89.00, $375.00
• Sizes: 10 mg, 50 mg
• Cas Number: 111-58-0
• Chemical Name: (9Z)-N-(2-Hydroxyethyl)-9-octadecenamide
• Formula: C20H39NO2
• Molecular Weight: 325.53
• Purity: >99 %
• Description: Lipid mediator and analog of anandamide (Cat. No. 1339) that is involved in peripheral regulation of feeding. Selective GPR55 agonist (EC 50 values are 0.44, >30 and >30 μ M at GPR55, CB 1 and CB 2 respectively) and PPAR α agonist (EC 50 = 120 nM). Induces satiety through activation of PPAR α and is also a ceramidase inhibitor. Also endogenous agonist at the GPR119 receptor.

Product References

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An anorexic lipid mediator regulated by feeding. - An anorexic lipid mediator regulated by feeding.

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Oleylethanolamide regulates feeding and body weight through activation of the - Oleylethanolamide regulates feeding and body weight through activation of the

Fu J, Gaetani S, Oveisi F, Lo Verme J, Serrano A, Rodriguez De Fonseca F, Rosengarth A, Luecke H, Di Giacomo B, Tarzia G, Piomelli D. Nature. 2003 Sep 4;425(6953):90-3.

The orphan receptor GPR55 is a novel cannabinoid receptor. - The orphan receptor GPR55 is a novel cannabinoid receptor.

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