OMDM-2

• Supplier: Tocris Bioscience
• Catalog: 0934
• Prices: $89.00, $375.00
• Sizes: 5 mg, 25 mg
• Function Type: Inhibitor
• Cas Number: 616884-63-0
• Chemical Name: (9Z)-N-[1-((R)-4-Hydroxbenzyl)-2-hydroxyethyl]-9-octadecenamide
• Formula: C27H45NO3
• Molecular Weight: 431.66
• Purity: >99 %
• Description: Metabolically stable inhibitor of anandamide cellular uptake (K i = 3 μ M). Displays relatively low affinity for CB 1 and CB 2 receptors (K i values are 5.1 and > 10 μ M) and for vanilloid VR1 receptors (EC 50 = 10 μ M). Has minimal activity against FAAH (K i > 50 μ M). Active in vivo .

Product References

Novel selective and metabolically stable inhibitors of anandamide cellular - Novel selective and metabolically stable inhibitors of anandamide cellular

Ortar G, Ligresti A, De Petrocellis L, Morera E, Di Marzo V. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

In vivo pharmacological actions of two novel inhibitors of anandamide cellular - In vivo pharmacological actions of two novel inhibitors of anandamide cellular

de Lago E, Ligresti A, Ortar G, Morera E, Cabranes A, Pryce G, Bifulco M, Baker D, Fernandez-Ruiz J, Di Marzo V. Eur J Pharmacol. 2004 Jan 26;484(2-3):249-57.