| Name | PEPA |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 1596 |
| Prices | $149.00, $629.00 |
| Sizes | 10 mg, 50 mg |
| Cas Number | 141286-78-4 |
| Chemical Name | 2-[2,6-Difluoro-4-[[2-[(phenylsulfonyl)amino]ethyl]thio]phenoxy]acetamide |
| Formula | C16H16F2N2O4S2 |
| Molecular Weight | 402.44 |
| Purity | >99 % |
| Description | Novel allosteric potentiator of AMPA receptor desensitization. Slows the rate of onset of desensitization and potentiates steady-state equilibrium currents induced by glutamate with subunit (GluR3/4 > GluR1) and splice variant (flop > flip) selectivity. Ameliorates post-ischemic memory impairment in rats following i.v. administration. |
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