| Name | PF 04885614 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4820 |
| Prices | $175.00, $709.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Chemical Name | 1-Methyl-[1-[4-(4-trifluoromethoxy)phenyl]-imidazol-2-yl]-ethanamine |
| Formula | C13H14F3N3O |
| Molecular Weight | 285.26 |
| Purity | >98 % |
| Description | Potent Na V 1.8 inhibitor (IC 50 = 53 nM for human Na V 1.8 channel). Exhibits selectivity for hNa V 1.8 over hNa V 1.6, hNa V 1.7, hNa V 1.1, hNa V 1.2 and hNa V 1.5 (IC 50 values are 4.2, 7.0, 11, 16 and 27 μ M respectively). Orally bioavailable. |
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