| Name | PFI 4 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 5072 |
| Prices | $209.00, $879.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 900305-37-5 |
| Chemical Name | N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-pyrrolidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide |
| Formula | C21H24N4O3 |
| Molecular Weight | 380.44 |
| Purity | >99 % |
| Description | Potent and selective BRPF1 bromodomain inhibitor (IC 50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of other bromodomains including BRPF2 (BRD1), BRPF3 and BRD4. Disrupts BRPF1 binding to histone H3.3. Cell permeable. |
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