Name | PHP 501 trifluoroacetate |
---|---|
Supplier | Tocris Bioscience |
Catalog | 0238 |
Prices | $225.00, $925.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 1236105-75-1 |
Chemical Name | 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidinetrifluoroacetate |
Formula | C20H21N3O.CF3CO2H |
Molecular Weight | 433.42 |
Purity | >98 % |
Description | Potent GABA A antagonist (K i = 0.0028 μ M at rat GABA A receptors; IC 50 = 0.024 μ M at human α 1 β 2 γ 2 GABA A -expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters. |
Supplier Page | Shop |