PHP 501 trifluoroacetate

Name PHP 501 trifluoroacetate
Supplier Tocris Bioscience
Catalog 0238
Prices $225.00, $925.00
Sizes 10 mg, 50 mg
Function Type Antagonist
Cas Number 1236105-75-1
Chemical Name 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidinetrifluoroacetate
Formula C20H21N3O.CF3CO2H
Molecular Weight 433.42
Purity >98 %
Description Potent GABA A antagonist (K i = 0.0028 μ M at rat GABA A receptors; IC 50 = 0.024 μ M at human α 1 β 2 γ 2 GABA A -expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.
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