PL 017

Name PL 017
Supplier Tocris Bioscience
Catalog 5338
Prices $65.00
Sizes 1 mg
Function Type Agonist
Cas Number 83397-56-2
Formula C29H37N5O5
Molecular Weight 535.64
Description Selective μ opioid receptor agonist (IC 50 values are 5.5 and > 10000 nM for inhibition of 125 I-FK 33,824 and 125 I-DADLE binding to μ and δ sites respectively). Produces naloxone-reversible analgesia, catalepsy and hyperthermia following central administration in rats in vivo .
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Product References

Potent morphiceptin analogs: structure activity relationships and morphine-like - Potent morphiceptin analogs: structure activity relationships and morphine-like

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Behavioral effects of the mu-opioid peptide agonists DAMGO, DALDA, and PL017 on - Behavioral effects of the mu-opioid peptide agonists DAMGO, DALDA, and PL017 on

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Body temperature and analgesic effects of selective mu and kappa opioid receptor - Body temperature and analgesic effects of selective mu and kappa opioid receptor

Xin L, Geller EB, Adler MW. J Pharmacol Exp Ther. 1997 Apr;281(1):499-507.