Name | PMX 205 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 4486 |
Prices | $265.00 |
Sizes | 1 mg |
Function Type | Antagonist |
Cas Number | 514814-49-4 |
Formula | C45H62N10O6 |
Molecular Weight | 839.05 |
Description | Potent C5a receptor peptide antagonist (IC 50 = 31 nM). Ameliorates experimentally-induced colon inflammation in mice. Reduces fibrillar amyloid deposits, decreases hyperphosphorylated tau levels and rescues cognitive function in a mouse model of Alzheimer's Disease. Orally active and brain penetrant. |
Supplier Page | Shop |
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