PSB 0739

• Supplier: Tocris Bioscience
• Catalog: 2573
• Prices: $175.00, $709.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 1052087-90-7
• Chemical Name: 1-Amino-9,10-dihydro-9,10-dioxo-4-[[4-(phenylamino)-3-sulfophenyl]amino]-2-anthracenesulfonicacidsodiumsalt
• Formula: C26H17N3Na2O8S2
• Molecular Weight: 609.54
• Purity: >95 %
• Description: Highly potent P2Y 12 receptor antagonist (K i = 24.9 nM). Unlike clopidogrel (Cat. No. 2490), does not require bioactivation.

Product References

High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 - High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12

Baqi Y, Atzler K, Kose M, Glanzel M, Muller CE. J Med Chem. 2009 Jun 25;52(12):3784-93.

Interaction of new, very potent non-nucleotide antagonists with Arg256 of the - Interaction of new, very potent non-nucleotide antagonists with Arg256 of the

Hoffmann K, Baqi Y, Morena MS, Glanzel M, Muller CE, von Kugelgen I. J Pharmacol Exp Ther. 2009 Nov;331(2):648-55.

Development of a comprehensive set of P2 receptor pharmacological research - Development of a comprehensive set of P2 receptor pharmacological research

Felix RA, Martin S, Pinion S, Crawford DJ. Purinergic Signal. 2012 Feb;8(Suppl 1):101-12.